SCHEMBL2977679

SCHEMBL2977679

C=Cc1ccnc(-c2ccccc2)c1C#N

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ADORA1 P30542 14/20 0.44
ADORA2A P29274 12/20 0.44
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
CRHBP P24387 1/20 0.40
RAB9A P51151 1/20 0.40
CRHR2 Q13324 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HPGD P15428 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2979399 0.85 ADORA2A (0.48) ALDH1A1MEN1KMT2ACYP1A2ADORA1
SCHEMBL2974174 0.81 SQOR (0.39) ALDH1A1MEN1KMT2ACYP1A2NPC1
SCHEMBL5671301 0.79 ALDH1A1 (0.41) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL7219981 0.76 ALDH1A1 (0.61) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL554431 0.76 PTGS1 (0.38) ALDH1A1KMT2AL3MBTL1NPC1MAPT
SCHEMBL5329331 0.75 ADORA1 (0.56) ADORA1ADORA2AHSD17B10
SCHEMBL15748249 0.73 MEN1 (0.35) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL30679309 0.73 PRKACA (0.36) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL398500 0.72 PTGS1 (0.39) ALDH1A1MAPTHSD17B10
SCHEMBL24311363 0.71 ALDH1A1 (0.45) ALDH1A1MEN1KMT2ACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229377-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP claimed
WO-2009076602-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO claimed