SCHEMBL7220451

SCHEMBL7220451

Cc1nc(-c2cccc(C#N)c2)c(CCl)s1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.43
ADORA1 P30542 5/20 0.43
ADORA2B P29275 3/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
CLK4 Q9HAZ1 1/20 0.41
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
GRM5 P41594 1/20 0.40
CFTR P13569 1/20 0.40
F11 P03951 1/20 0.39
PIN1 Q13526 1/20 0.39
ADORA3 P0DMS8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6287392 0.75 F11 (0.52) ADORA2AADORA1ADORA2BPTGDR2GRM5
SCHEMBL6283502 0.73 ADORA2A (0.45) ADORA2AADORA1ADORA2BPTGDR2GRM5
SCHEMBL8205342 0.73 CDK4 (0.54) ADORA2AADORA1ADORA2BCLK4CTSS
SCHEMBL7430278 0.70 IDO1 (0.43) CLK4F11PIN1
SCHEMBL5510284 0.69 PTGS2 (0.51) PTGDR2
SCHEMBL4854539 0.68 PPARG (0.47) ADORA2AADORA1ADORA2BCLK4CTSS
SCHEMBL12636667 0.67 PRF1 (0.50) ADORA2AADORA1ADORA2BCLK4CTSS
SCHEMBL6237896 0.67 ADORA2A (0.51) ADORA2AADORA1ADORA2BCLK4CFTR
SCHEMBL24763023 0.67 ADORA1 (0.58) ADORA2AADORA1ADORA2BCLK4CFTR
SCHEMBL19169352 0.67 ADORA2A (0.59) ADORA2AADORA1ADORA2BCLK4CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6534535-B1 Administering indole derivative as anticoagulant MILLENNIUM PHARMACEUTICALS, INC. 2003-03-18 US disclosed
WO-2001012600-A9 INHIBITORS OF FACTOR Xa COR THERAPEUTICS INC (US) 2002-09-12 WO disclosed
WO-2001012600-A1 INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2001-02-22 WO disclosed