SCHEMBL7430278

SCHEMBL7430278

Cc1n[nH]c(CCl)c1-c1cccc(C#N)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.43
MAP4K4 O95819 1/20 0.41
GSK3A P49840 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
MAOB P27338 1/20 0.40
FASN P49327 1/20 0.39
PGR P06401 2/20 0.39
F11 P03951 1/20 0.39
PIN1 Q13526 1/20 0.39
AR P10275 1/20 0.39
LRRK2 Q5S007 1/20 0.39
GRK6 P43250 1/20 0.39
PIK3R1 P27986 2/20 0.39
PIK3CA P42336 2/20 0.39
DHFR P00374 1/20 0.38
CNR2 P34972 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7395177 0.79 IDO1 (0.46) IDO1MAP4K4GSK3ACLK4MAOB
SCHEMBL30239372 0.75 CHEK1 (0.57) IDO1MAP4K4GSK3ACLK4MAOB
SCHEMBL24963400 0.75 CHEK1 (0.57) IDO1MAP4K4GSK3ACLK4MAOB
SCHEMBL7404293 0.75 F11 (0.52) IDO1MAP4K4GSK3ACLK4FASN
SCHEMBL7220451 0.70 ADORA2A (0.43) CLK4F11PIN1
SCHEMBL16905206 0.69 CLK4 (0.52) IDO1MAP4K4CLK4MAOBPGR
SCHEMBL8807143 0.68 IDO1 (0.53) IDO1MAP4K4GSK3ACLK4MAOB
SCHEMBL5269506 0.68 L3MBTL1 (0.59) IDO1MAP4K4GSK3ACLK4MAOB
SCHEMBL8205342 0.67 CDK4 (0.54) IDO1CLK4MAOBF11PIN1
SCHEMBL27518736 0.67 LRRK2 (0.49) IDO1CLK4MAOBPGRF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001012600-A9 INHIBITORS OF FACTOR Xa COR THERAPEUTICS INC (US) 2002-09-12 WO disclosed
WO-2001012600-A1 INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2001-02-22 WO disclosed