SCHEMBL7220496

SCHEMBL7220496

Cc1ccc(-c2cncc(C=CC(=O)NC3CCC(CN(C)C4CCOCC4)CC3)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.41
CCR2 P41597 2/20 0.39
ALDH1A1 P00352 3/20 0.37
RAB9A P51151 3/20 0.36
NPC1 O15118 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
DRD3 P35462 3/20 0.35
DRD2 P14416 2/20 0.35
GRIN2B Q13224 1/20 0.35
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
ITGA5 P08648 1/20 0.34
GABRA5 P31644 1/20 0.34
LMNA P02545 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7220493 1.00 HDAC1 (0.41) HDAC1CCR2ALDH1A1RAB9ANPC1
SCHEMBL7224635 0.83 ALDH1A1 (0.37) CCR2ALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL7219091 0.83 CCR2 (0.37) CCR2ALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL7224629 0.83 ALDH1A1 (0.37) CCR2ALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL7219085 0.83 CCR2 (0.37) CCR2ALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL5210797 0.80 CCR2 (0.55) HDAC1CCR2
SCHEMBL5210801 0.80 CCR2 (0.55) HDAC1CCR2
SCHEMBL7221605 0.72 OPRK1 (0.40) CCR2ALDH1A1GABRA5
SCHEMBL7221600 0.72 OPRK1 (0.40) CCR2ALDH1A1GABRA5
SCHEMBL8436676 0.70 C3AR1 (0.50) ALDH1A1RAB9ANPC1SMN1; SMN2CCNC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627651-B1 Exhibiting preventive and therapeutic effects against HIV infectious diseases wherein R1 is an optionally substituted five- or six-membered ring group; X1 is a free valency or the like; W is a divalent group and inhibitors of HIV (human TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-30 US disclosed
EP-1182195-A1 CYCLIC COMPOUNDS AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-27 EP disclosed