SCHEMBL7220659

SCHEMBL7220659

COc1ccc(CC2(C)NC(C)OC2=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.44
GLA P06280 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
TLR9 Q9NR96 1/20 0.42
MMP2 P08253 4/20 0.40
MMP9 P14780 4/20 0.40
MMP8 P22894 4/20 0.40
MMP13 P45452 4/20 0.40
GRM2 Q14416 1/20 0.39
DAO P14920 3/20 0.39
LMNA P02545 1/20 0.39
CMA1 P23946 1/20 0.38
CRBN Q96SW2 1/20 0.37
GAA P10253 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL542639 0.71 SMN1; SMN2 (0.73) NPSR1SMN1; SMN2MMP2MMP9MMP8
SCHEMBL15569546 0.69 NPSR1 (0.56) NPSR1GLASMN1; SMN2TLR9MMP2
SCHEMBL5443745 0.66 MMP2 (0.70) NPSR1SMN1; SMN2MMP2MMP9MMP8
SCHEMBL13651912 0.66 GLA (0.42) NPSR1GLASMN1; SMN2TLR9LMNA
SCHEMBL7220662 0.65 NPSR1 (0.41) NPSR1GLASMN1; SMN2TLR9MMP2
SCHEMBL29002709 0.65 GLA (0.44) NPSR1GLASMN1; SMN2GRM2ALDH1A1
SCHEMBL8515475 0.64 GLA (0.40) NPSR1GLASMN1; SMN2MMP2MMP9
SCHEMBL10590941 0.64 LDHA (0.46) NPSR1GLASMN1; SMN2TLR9ALDH1A1
SCHEMBL19559791 0.64 MMP2 (0.45) NPSR1GLASMN1; SMN2MMP2MMP9
SCHEMBL1603072 0.63 HSD11B1 (0.49) NPSR1GLASMN1; SMN2CRBNGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6504046-B1 Cyclization of nitriles using acids, to form oxazolinone chemical intermediates such as 2-phenyl-4-isopropyl-4-methyl-1,3-oxazol-5-one, used as fungicides IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2003-01-07 US disclosed
EP-1092705-A1 PROCESS FOR THE PREPARATION OF AMIDES IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 2001-04-18 EP disclosed