SCHEMBL7222633

SCHEMBL7222633

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(Oc2ccccc2NS(=O)(=O)C(F)(F)F)s1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 1/20 0.33
PTGS1 P23219 3/20 0.32
PTGS2 P35354 3/20 0.32
PRKCB P05771 2/20 0.32
PRKCA P17252 2/20 0.32
PRKCE Q02156 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CXCR2 P25025 1/20 0.32
CHRNA7 P36544 1/20 0.31
PTK2 Q05397 1/20 0.31
IDO1 P14902 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7229598 0.89 ALDH1A1 (0.42) MRGPRX1KDM4EALDH1A1HPGDTSHR
SCHEMBL7224864 0.86 ANO1 (0.35) MRGPRX1PRKCBCXCR2CHRNA7
SCHEMBL7233624 0.85 KDM1A (0.33) PTGS1PTGS2PRKCBPRKCAPRKCE
SCHEMBL7232823 0.85 EPHX2 (0.36) CHRNA7
SCHEMBL7233645 0.84 PTPN1 (0.42) PTK2CA2
SCHEMBL7225638 0.84 SMN1; SMN2 (0.36) ALDH1A1CXCR2CHRNA7
SCHEMBL7224194 0.83 CHRNA7 (0.35) CHRNA7
SCHEMBL7233015 0.83 CHRNA7 (0.39) PRKCBPRKCAPRKCEKDM4EALDH1A1
SCHEMBL7232082 0.82 CXCR2 (0.34) MRGPRX1ALDH1A1CXCR2CHRNA7
SCHEMBL7230631 0.81 CHRNA7 (0.33) CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed