SCHEMBL7224864

SCHEMBL7224864

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(Oc2ccccc2NC(=O)C(F)(F)F)s1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ANO1 Q5XXA6 2/20 0.35
CXCR2 P25025 1/20 0.33
MRGPRX1 Q96LB2 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
CHRNA7 P36544 1/20 0.32
GAA P10253 1/20 0.31
PKM P14618 1/20 0.31
PDK1 Q15118 1/20 0.31
PDK2 Q15119 1/20 0.31
PDK3 Q15120 1/20 0.31
PDK4 Q16654 1/20 0.31
JAK2 O60674 1/20 0.31
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
KLK7 P49862 1/20 0.31
SLC6A3 Q01959 2/20 0.30
PRKCB P05771 1/20 0.30
PRKCD Q05655 1/20 0.30
MLYCD O95822 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7225638 0.89 SMN1; SMN2 (0.36) CXCR2SMN1; SMN2CHRNA7GAAPKM
SCHEMBL7232082 0.88 CXCR2 (0.34) CXCR2MRGPRX1SMN1; SMN2CHRNA7GAA
SCHEMBL7232823 0.86 EPHX2 (0.36) CHRNA7SLC6A3
SCHEMBL7222633 0.86 MRGPRX1 (0.33) CXCR2MRGPRX1CHRNA7PRKCB
SCHEMBL7231099 0.84 L3MBTL1 (0.34) SMN1; SMN2PDK1PDK2PDK3PDK4
SCHEMBL7229598 0.84 ALDH1A1 (0.42) CXCR2MRGPRX1CHRNA7
SCHEMBL7222908 0.84 EPHX2 (0.34) SMN1; SMN2PDK1PDK2PDK3PDK4
SCHEMBL7224194 0.83 CHRNA7 (0.35) CHRNA7SLC6A3
SCHEMBL7223114 0.83 CHRNA7 (0.40) SMN1; SMN2CHRNA7TP53MAPT
SCHEMBL7223853 0.82 CHRNA7 (0.43) SMN1; SMN2CHRNA7SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed