SCHEMBL7223178

SCHEMBL7223178

CC(=O)Nc1c(Br)cc(Br)cc1C(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
GAA P10253 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
KCNJ11 Q14654 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.36
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
MAPT P10636 2/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
RXFP1 Q9HBX9 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPK14 Q16539 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7224249 0.85 ALDH1A1 (0.45) ALDH1A1GAATDP1KCNJ11PTGS1
SCHEMBL6354671 0.83 ALDH1A1 (0.44) ALDH1A1TDP1KCNJ11MAPTCA1
SCHEMBL31218457 0.77 ALDH1A1 (0.45) ALDH1A1KCNJ11MAPTCA1CA2
SCHEMBL21979989 0.77 ALDH1A1 (0.45) ALDH1A1KCNJ11MAPTCA1CA2
SCHEMBL25096707 0.75 ALDH1A1 (0.42) ALDH1A1KCNJ11MAPTCA1CA2
SCHEMBL7223876 0.74 ALDH1A1 (0.52) ALDH1A1GAATDP1KCNJ11PTGS1
SCHEMBL7224330 0.74 ALDH1A1 (0.72) ALDH1A1GAATDP1PTGS1PTGS2
SCHEMBL8528629 0.74 AKR1C3 (0.52) ALDH1A1PTGS1MAPTMEN1KMT2A
SCHEMBL31210947 0.72 ALOX15 (0.47) ALDH1A1MAPTMEN1KMT2A
SCHEMBL27899868 0.72 ALDH1A1 (0.37) ALDH1A1KCNJ11MAPTCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6521603-B2 Amide, thioamide, amidine and thioester derivatives containing a benzene, pyridine, thiophene, furan, pyrrole, pyrazole, thiazole or isothiazole ring MONSANTO TECHNOLOGY LLC 2003-02-18 US claimed