SCHEMBL7224766

SCHEMBL7224766

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1cnc(-c2ccccn2)s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
CHRNA7 P36544 2/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
USP30 Q70CQ3 1/20 0.39
CYP3A4 P08684 1/20 0.38
BCAT2 O15382 2/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7071274 0.86 USP30 (0.53) ALDH1A1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL7232138 0.86 USP30 (0.36) ALDH1A1CHRNA7USP30
SCHEMBL7224345 0.85 CHRNA7 (0.60) CHRNA7NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL374986 0.85 CHRNA7 (0.60) CHRNA7NPC1MAPTRAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL7075524 0.85 USP30 (0.52) ALDH1A1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL7234885 0.85 GSK3B (0.35) CHRNA7USP30
SCHEMBL7226932 0.84 SLC6A3 (0.37) CHRNA7USP30HDAC3HDAC4HDAC1
Hydrochloric Acid SCHEMBL7231896 0.84 CHRNA7 (0.59) CHRNA7NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL7075331 0.83 USP30 (0.39) ALDH1A1NPC1RAB9ASMN1; SMN2USP30
SCHEMBL7234311 0.83 USP30 (0.39) NPC1RAB9AUSP30HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed