SCHEMBL7224779

SCHEMBL7224779

C#CCOc1cc(NC(=O)N(N)CCO)c(F)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.36
MAOA P21397 2/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
PGK1 P00558 1/20 0.34
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34
CYP2B6 P20813 1/20 0.33
MAOB P27338 2/20 0.33
DHODH Q02127 6/20 0.32
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
MAPT P10636 2/20 0.31
LIMK1 P53667 1/20 0.31
NR4A1 P22736 1/20 0.31
NR4A2 P43354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19048790 0.87 LMNA (0.36) LMNAMAOAHDAC1HDAC2HDAC8
SCHEMBL16774420 0.87 ALDH1A1 (0.36) LMNAMAOAHDAC1HDAC2HDAC8
SCHEMBL7253923 0.84 LMNA (0.36) LMNAMAOAHDAC1HDAC2HDAC8
SCHEMBL7249853 0.83 POLB (0.44) LMNATSHRMAPT
SCHEMBL17197232 0.81 LMNA (0.41) LMNAMAOAHDAC1HDAC2HDAC8
SCHEMBL8982258 0.78 NPC1 (0.46) LMNAMAOAHDAC1HDAC2HDAC8
SCHEMBL8998078 0.78 CYP2B6 (0.44) LMNAMAOAHDAC1HDAC2HDAC8
SCHEMBL16774399 0.77 DHODH (0.45) LMNAMAOAHDAC1HDAC2HDAC8
SCHEMBL16774378 0.77 PGK1 (0.41) LMNAMAOAHDAC1HDAC2HDAC8
SCHEMBL16774525 0.76 PGK1 (0.39) LMNAMAOAHDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6639070-B1 4-substituted 1,3,4-oxadiazines; herbicides BASF AKTIENGESELLSCHAFT (DE) 2003-10-28 US disclosed
US-6525000-B1 N-aminoureas are reacted with formaldehyde to give methyleneimino ureas, cyclizing these to give tetrahydro-4H-1,3,4-oxa(or thia)diazines, and cyclizing the fused triazoles using phosgene; herbicides BASF AKTIENGESELLSCHAFT (DE) 2003-02-25 US disclosed