SCHEMBL7225022

SCHEMBL7225022

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(-c2ccc(Oc3ccccc3)cc2)o1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 4/20 0.40
MAPT P10636 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
ABCB1 P08183 1/20 0.40
POLB P06746 1/20 0.40
PTPN1 P18031 1/20 0.40
PTPN11 Q06124 1/20 0.40
MMP13 P45452 2/20 0.39
MMP2 P08253 1/20 0.39
MMP7 P09237 1/20 0.39
MMP9 P14780 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 2/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL375394 0.91 NPC1 (0.44) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL7074460 0.91 NPC1 (0.44) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL7230430 0.91 RAB9A (0.41) NPC1RAB9AALDH1A1KDM4EMAPT
Hydrochloric Acid SCHEMBL7075781 0.90 NPC1 (0.43) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL7233285 0.89 MMP13 (0.48) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL7225861 0.88 PTPN1 (0.45) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL7225621 0.87 NPC1 (0.41) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL7233288 0.86 NPC1 (0.46) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL7232127 0.86 SLC9A1 (0.48) NPC1RAB9AALDH1A1KDM4EMAPT
SCHEMBL7226086 0.86 SCN10A (0.50) NPC1RAB9AL3MBTL1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed