SCHEMBL7225191

SCHEMBL7225191

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1cnc(-c2ccncc2F)s1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 5/20 0.35
ADORA2A P29274 3/20 0.35
ADORA1 P30542 1/20 0.35
PIM1 P11309 3/20 0.34
PIM3 Q86V86 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
CYP3A4 P08684 3/20 0.34
CYP2C19 P33261 3/20 0.34
USP30 Q70CQ3 1/20 0.34
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32
SLC6A3 Q01959 1/20 0.32
KDM1A O60341 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
ADORA3 P0DMS8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7234785 0.94 PIM1 (0.34) PIM1PIM3PIM2USP30CHRNB2
SCHEMBL7075331 0.89 USP30 (0.39) PIM1PIM3USP30CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL7077995 0.88 USP30 (0.39) PIM1PIM3USP30CHRNB2CHRNA4
SCHEMBL7227071 0.86 HDAC3 (0.44) CHRNB2CHRNA4SLC6A3
SCHEMBL7225497 0.86 HDAC3 (0.37) PIM1CHRNB2CHRNA4SLC6A3
SCHEMBL7223173 0.85 CDC7 (0.43) CYP3A4USP30SLC6A3
SCHEMBL7223374 0.84 CHRNB2 (0.36) USP30CHRNB2CHRNA4
SCHEMBL7233042 0.84 USP30 (0.36) PIM1PIM3PIM2USP30CHRNB2
SCHEMBL7223521 0.83 PIM1 (0.39) PIM1PIM3PIM2USP30CHRNB2
SCHEMBL7225628 0.82 USP30 (0.36) PIM1PIM3PIM2USP30CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed