SCHEMBL7225311

SCHEMBL7225311

C=C(CN1CCNCC1)CN1CCNC1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 2/20 0.39
CHRM3 P20309 2/20 0.39
SIGMAR1 Q99720 6/20 0.36
SMN1; SMN2 Q16637 3/20 0.34
ALDH1A1 P00352 1/20 0.34
STAT6 P42226 1/20 0.34
POLB P06746 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CXCR4 P61073 2/20 0.32
KDM5C P41229 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
EGFR P00533 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7223824 0.96 CHRM5 (0.33) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL7230790 0.92 CHRM5 (0.37) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL7222024 0.91 CHRM5 (0.44) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL7230380 0.90 SIGMAR1 (0.37) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL7224032 0.87 KDM4E (0.40) CHRM5CHRM3SMN1; SMN2ALDH1A1HSD17B10
SCHEMBL7694509 0.84 CHRM5 (0.44) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL7222004 0.83 SIGMAR1 (0.43) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL1400999 0.80
SCHEMBL7230900 0.79 CHRM5 (0.41) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL7230894 0.79 CHRM5 (0.41) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6552226-B1 Rapid; low temperature; one pot synthesis; reduced catalytic quantities of such as lewis acid and tertiary amine; entiomerically pure products THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2003-04-22 US disclosed
WO-2002026683-A1 TANDEM ACYL-CLAISEN REARRANGEMENT IN THE PREPARATION OF CHIRAL PRODUCTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2002-04-04 WO disclosed