SCHEMBL7222004

SCHEMBL7222004

C=C(CN1CCCCC1)CN1CCNCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.43
CHRM5 P08912 2/20 0.43
CHRM3 P20309 2/20 0.43
CXCR4 P61073 7/20 0.41
GAA P10253 1/20 0.39
CA2 P00918 1/20 0.39
CHKA P35790 1/20 0.39
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
ADRA2C P18825 1/20 0.36
CCR2 P41597 1/20 0.36
CXCL12 P48061 1/20 0.36
BLM P54132 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
RAD52 P43351 1/20 0.35
STAT6 P42226 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7694509 0.98 CHRM5 (0.44) SIGMAR1CHRM5CHRM3CXCR4GAA
SCHEMBL7222024 0.91 CHRM5 (0.44) SIGMAR1CHRM5CHRM3CXCR4ALDH1A1
SCHEMBL7230380 0.90 SIGMAR1 (0.37) SIGMAR1CHRM5CHRM3CXCR4GAA
SCHEMBL7230790 0.88 CHRM5 (0.37) SIGMAR1CHRM5CHRM3CXCR4GAA
SCHEMBL7222432 0.86 GAA (0.48) CHRM5GAAALDH1A1MEN1ADRA2C
SCHEMBL7221817 0.86 GAA (0.48) CHRM5GAAALDH1A1MEN1ADRA2C
SCHEMBL7228369 0.83 ALDH1A1 (0.46) GAAALDH1A1MEN1KMT2AHRH3
SCHEMBL7225311 0.83 CHRM5 (0.39) SIGMAR1CHRM5CHRM3CXCR4ALDH1A1
SCHEMBL7231084 0.79 KDM4E (0.44) SIGMAR1CHRM5CHRM3ALDH1A1SMN1; SMN2
SCHEMBL7222798 0.79 CHRM5 (0.44) SIGMAR1CHRM5CHRM3CXCR4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6552226-B1 Rapid; low temperature; one pot synthesis; reduced catalytic quantities of such as lewis acid and tertiary amine; entiomerically pure products THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2003-04-22 US disclosed
WO-2002026683-A1 TANDEM ACYL-CLAISEN REARRANGEMENT IN THE PREPARATION OF CHIRAL PRODUCTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2002-04-04 WO disclosed