SCHEMBL7225473

SCHEMBL7225473

CNc1ccccc1-c1ncc(C(=O)N[C@@H]2C[C@H]3CC[C@@H]2N3)s1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK11 Q15759 1/20 0.42
MAPK14 Q16539 1/20 0.42
USP30 Q70CQ3 1/20 0.39
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36
ACHE P22303 3/20 0.35
MAOA P21397 1/20 0.34
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7224115 0.90 MAPK11 (0.43) MAPK11MAPK14USP30HTR3EHTR3B
SCHEMBL7231132 0.89 MAPK11 (0.42) MAPK11MAPK14USP30HTR3EHTR3B
SCHEMBL7226023 0.88 USP30 (0.41) MAPK11MAPK14USP30HTR3EHTR3B
SCHEMBL7225952 0.88 MAPK14 (0.45) MAPK11MAPK14USP30HTR3EHTR3B
SCHEMBL7234311 0.87 USP30 (0.39) MAPK11MAPK14USP30HTR3EHTR3B
SCHEMBL7075331 0.87 USP30 (0.39) MAPK11MAPK14USP30HTR3EHTR3B
SCHEMBL7223360 0.86 MAPK11 (0.39) MAPK11MAPK14USP30HTR3EHTR3B
Hydrochloric Acid SCHEMBL7077995 0.86 USP30 (0.39) MAPK11MAPK14USP30HTR3EHTR3B
SCHEMBL7233186 0.86 USP30 (0.39) MAPK11MAPK14USP30HTR3EHTR3B
SCHEMBL7230337 0.86 MAPK11 (0.49) MAPK11MAPK14USP30HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed