SCHEMBL7225952

SCHEMBL7225952

Cc1ccccc1-c1ncc(C(=O)N[C@@H]2C[C@H]3CC[C@@H]2N3)s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.45
MAPK11 Q15759 2/20 0.45
USP30 Q70CQ3 1/20 0.41
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
RIPK2 O43353 1/20 0.35
LCK P06239 3/20 0.35
MAPK13 O15264 1/20 0.35
EGFR P00533 1/20 0.35
FYN P06241 1/20 0.35
HCK P08631 1/20 0.35
SRC P12931 1/20 0.35
JAK3 P52333 1/20 0.35
MAPK12 P53778 1/20 0.35
ALDH1A1 P00352 1/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7226023 0.90 USP30 (0.41) MAPK14MAPK11USP30HTR3EHTR3B
SCHEMBL7234311 0.89 USP30 (0.39) MAPK14MAPK11USP30HTR3EHTR3B
SCHEMBL7075331 0.89 USP30 (0.39) MAPK14MAPK11USP30HTR3EHTR3B
SCHEMBL7225473 0.88 MAPK11 (0.42) MAPK14MAPK11USP30HTR3EHTR3B
SCHEMBL7230337 0.88 MAPK11 (0.49) MAPK14MAPK11USP30HTR3EHTR3B
SCHEMBL7233186 0.88 USP30 (0.39) MAPK14MAPK11USP30HTR3EHTR3B
Hydrochloric Acid SCHEMBL7077995 0.88 USP30 (0.39) MAPK14MAPK11USP30HTR3EHTR3B
SCHEMBL7233270 0.87 HDAC3 (0.48) MAPK14MAPK11USP30HTR3EHTR3B
SCHEMBL7224115 0.86 MAPK11 (0.43) MAPK14MAPK11USP30HTR3EHTR3B
SCHEMBL7231086 0.85 USP30 (0.43) MAPK14MAPK11USP30HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed