SCHEMBL7225783

SCHEMBL7225783

O=C(O)[C@@H](OS(=O)(=O)C(F)(F)F)C1CCCCC1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.37
DPP4 P27487 1/20 0.33
ALDH1A1 P00352 1/20 0.32
MMP1 P03956 1/20 0.32
MMP2 P08253 1/20 0.32
MMP3 P08254 1/20 0.32
MMP7 P09237 1/20 0.32
MMP13 P45452 1/20 0.32
PDK1 Q15118 1/20 0.30
PDK2 Q15119 1/20 0.30
PDK3 Q15120 1/20 0.30
PDK4 Q16654 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4740510 1.00 EPHX1 (0.37) EPHX1DPP4ALDH1A1MMP1MMP2
SCHEMBL1614329 0.77 EPHX1 (0.32) EPHX1
SCHEMBL18706685 0.75 EPHX1 (0.31) EPHX1
SCHEMBL1064167 0.74
SCHEMBL32677608 0.73 CYP3A4 (0.48) EPHX1DPP4ALDH1A1
SCHEMBL32677609 0.73 CYP3A4 (0.48) EPHX1DPP4ALDH1A1
SCHEMBL26349710 0.73 CYP3A4 (0.48) EPHX1DPP4ALDH1A1
SCHEMBL31355393 0.73 EPHX1 (0.43) EPHX1DPP4ALDH1A1
SCHEMBL22609005 0.72 SLC1A3 (0.36) MMP1MMP2MMP3MMP13
SCHEMBL22609004 0.72 SLC1A3 (0.36) MMP1MMP2MMP3MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6531484-B2 Viricides for preventing infection by HIV, treating infection by HIV, delaying of the onset of AIDS, or treating AIDS MERCK & CO., INC. 2003-03-11 US disclosed
US-20020198178-A1 Pyrrolidine modulators of CCR5 chemokine receptor activity MERCK SHARP & DOHME CORP. 2002-12-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020198178-A1 Pyrrolidine modulators of CCR5 chemokine receptor activity CCR5, CCR1, CCL5 EPHX1 3785/4885DPP4 3549/4885ALDH1A1 3312/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.