SCHEMBL7225896

SCHEMBL7225896

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ncc(-c2cc(F)cc(F)c2)o1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
ACKR3 P25106 4/20 0.37
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
SLC6A3 Q01959 3/20 0.34
CHRNB2 P17787 2/20 0.34
CHRNA4 P43681 2/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
ITGA5 P08648 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRND Q07001 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7230444 0.91 CA12 (0.39) CA12CA1CA2CA4ACKR3
SCHEMBL7234886 0.90 FAAH (0.46) CA12CA1CA2CA4ACKR3
SCHEMBL7226619 0.89 HDAC1 (0.46) CA12CA1CA2CA4ACKR3
SCHEMBL7231176 0.87 CA12 (0.39) CA12CA1CA2CA4HDAC1
SCHEMBL7233445 0.87 CA12 (0.41) CA12CA1CA2CA4ACKR3
SCHEMBL7233239 0.87 CA12 (0.39) CA12CA1CA2CA4ACKR3
SCHEMBL7231627 0.86 CA12 (0.42) CA12CA1CA2CA4ACKR3
SCHEMBL7073214 0.85 TUBB4A (0.47) CA12CA1CA2CA4HDAC1
Hydrochloric Acid SCHEMBL7072564 0.84 TUBB4A (0.46) CA12CA1CA2CA4HDAC1
SCHEMBL7234556 0.84 CA12 (0.44) CA12CA1CA2CA4ACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed