SCHEMBL7233239

SCHEMBL7233239

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ncc(-c2ccnc(F)c2)o1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
TAS1R2 Q8TE23 1/20 0.38
ACKR3 P25106 4/20 0.37
CSNK2A2 P19784 1/20 0.35
CSNK2A1 P68400 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
KDM1A O60341 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7233445 0.90 CA12 (0.41) CA12CA1CA2CA4ACKR3
SCHEMBL7234556 0.88 CA12 (0.44) CA12CA1CA2CA4ACKR3
SCHEMBL7234886 0.87 FAAH (0.46) CA12CA1CA2CA4ACKR3
SCHEMBL7226619 0.87 HDAC1 (0.46) CA12CA1CA2CA4ACKR3
SCHEMBL7225896 0.87 CA12 (0.39) CA12CA1CA2CA4ACKR3
SCHEMBL7231627 0.86 CA12 (0.42) CA12CA1CA2CA4ACKR3
SCHEMBL7230583 0.85 FAAH (0.44) CA12CA1CA2CA4ACKR3
SCHEMBL7223707 0.85 NPC1 (0.38) TAS1R3TAS1R1TAS1R2KDM1A
SCHEMBL7073214 0.84 TUBB4A (0.47) CA12CA1CA2CA4CHRNB2
SCHEMBL7231308 0.84 FAAH (0.45) CA12CA1CA2CA4CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed