SCHEMBL7226707

SCHEMBL7226707

O=C(C1CC1)N(CC1CCCN(CCc2ccccc2)C1)N1CCCCC1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
KMT2A Q03164 2/20 0.49
OPRM1 P35372 3/20 0.48
SIGMAR1 Q99720 1/20 0.46
LTA4H P09960 1/20 0.46
EPHX2 P34913 1/20 0.46
CHRNB2 P17787 1/20 0.46
CHRNB4 P30926 1/20 0.46
CHRNA3 P32297 1/20 0.46
CHRNA4 P43681 1/20 0.46
CCR2 P41597 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5870761 0.83 OPRM1 (0.50) KMT2AOPRM1SIGMAR1LTA4HEPHX2
SCHEMBL5871105 0.78 SMN1; SMN2 (0.53) KMT2AOPRM1LTA4HEPHX2CHRNB2
SCHEMBL5870735 0.76 CHRNB2 (0.46) KDM4EKMT2AOPRM1LTA4HEPHX2
SCHEMBL7226706 0.76 OPRM1 (0.51) KMT2AOPRM1CHRNB2CHRNB4CHRNA3
SCHEMBL5870682 0.75 OPRD1 (0.62) OPRM1SIGMAR1CHRNA4
SCHEMBL5870753 0.75 OPRD1 (0.62) OPRM1SIGMAR1CHRNA4
SCHEMBL5870685 0.75 OPRD1 (0.62) OPRM1SIGMAR1CHRNA4
SCHEMBL5870834 0.74 OPRM1 (0.55) OPRM1SIGMAR1CHRNA4
SCHEMBL5870832 0.74 OPRM1 (0.55) OPRM1SIGMAR1CHRNA4
SCHEMBL5870894 0.73 OPRD1 (0.49) KMT2AOPRM1CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6645980-B1 Ligands for biological receptors such as opiate receptors or G-protein coupled receptors used for treating pain, drug dependence or tinnitus in mammals SEPRACOR INC. 2003-11-11 US disclosed