SCHEMBL7226992

SCHEMBL7226992

O=C(O)[C@@H]1CNCCN1S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 14/20 0.50
ITGA4 P13612 14/20 0.50
ITGB7 P26010 1/20 0.47
MMP1 P03956 1/20 0.46
MMP3 P08254 1/20 0.46
MMP7 P09237 1/20 0.46
MMP9 P14780 1/20 0.46
MMP13 P45452 1/20 0.46
CNR1 P21554 2/20 0.42
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7226993 1.00 ITGB1 (0.50) ITGB1ITGA4ITGB7MMP1MMP3
Hydrochloric Acid SCHEMBL7454639 0.99 ITGB1 (0.49) ITGB1ITGA4ITGB7MMP1MMP3
SCHEMBL5201269 0.81 ITGB1 (0.58) ITGB1ITGA4ITGB7CNR1
SCHEMBL5201278 0.81 ITGB1 (0.58) ITGB1ITGA4ITGB7CNR1
SCHEMBL27488462 0.80 MMP9 (0.56) MMP1MMP3MMP7MMP9MMP13
SCHEMBL3904078 0.80 ITGB1 (0.67) ITGB1ITGA4ITGB7MMP13KDM4E
SCHEMBL3904073 0.80 ITGB1 (0.67) ITGB1ITGA4ITGB7MMP13KDM4E
SCHEMBL2988722 0.79 ITGB1 (0.66) ITGB1ITGA4ITGB7MMP13
SCHEMBL2988718 0.79 ITGB1 (0.66) ITGB1ITGA4ITGB7MMP13
SCHEMBL27583610 0.78 MMP1 (0.54) MMP1MMP3MMP7MMP9MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6645939-B1 Very late antigen-4 (VLA) integrin antagonists; antiallergens, antiasthmatics, and antiinflammatory agents; multiple sclerosis, autoimmune disease treatment MERCK & CO., INC. 2003-11-11 US disclosed