SCHEMBL7227405

SCHEMBL7227405

Cc1ccc(-c2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 2/20 0.50
MAPK12 P53778 2/20 0.50
MAPK11 Q15759 2/20 0.50
MAPK14 Q16539 2/20 0.50
ESR1 P03372 1/20 0.40
ESRRG P62508 1/20 0.40
ESR2 Q92731 1/20 0.40
PTPN1 P18031 1/20 0.40
PTPN11 Q06124 1/20 0.40
CHRNA7 P36544 7/20 0.39
HTR3E A5X5Y0 4/20 0.39
HTR3B O95264 4/20 0.39
HTR3A P46098 4/20 0.39
HTR3D Q70Z44 4/20 0.39
HTR3C Q8WXA8 4/20 0.39
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7223964 0.88 CHRNA7 (0.42) MAPK13MAPK12MAPK11MAPK14ESR1
SCHEMBL7243631 0.88 CHRNA7 (0.42) MAPK13MAPK12MAPK11MAPK14ESR1
SCHEMBL7243634 0.88 CHRNA7 (0.42) MAPK13MAPK12MAPK11MAPK14ESR1
SCHEMBL7224991 0.87 ESRRG (0.46) MAPK11MAPK14ESR1ESRRGESR2
SCHEMBL7224866 0.87 CTSC (0.40) MAPK13MAPK12MAPK11MAPK14ESR1
SCHEMBL7230436 0.86 CTSS (0.42) MAPK13MAPK12MAPK11MAPK14ESR1
SCHEMBL7224299 0.85 NPC1 (0.45) ESR1ESRRGESR2PTPN1PTPN11
SCHEMBL7232814 0.84 CHRNA7 (0.37) MAPK13MAPK12MAPK11MAPK14CHRNA7
SCHEMBL7231746 0.84 HDAC3 (0.56) MAPK13MAPK12MAPK11MAPK14CHRNA7
SCHEMBL7223147 0.83 HDAC1 (0.41) MAPK11MAPK14CHRNA7HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed