SCHEMBL7224866

SCHEMBL7224866

COc1ccc(-c2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSC P53634 1/20 0.40
KDM4E B2RXH2 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
ESR1 P03372 1/20 0.38
ESRRG P62508 1/20 0.38
ESR2 Q92731 1/20 0.38
PTPN1 P18031 1/20 0.38
PTPN11 Q06124 1/20 0.38
MAPK13 O15264 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
TEC P42680 1/20 0.38
TXK P42681 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7227405 0.87 MAPK13 (0.50) KDM4EALDH1A1GAAESR1ESRRG
SCHEMBL7230944 0.87 CTSS (0.44) CTSCMAPK13MAPK12MAPK11MAPK14
SCHEMBL7223964 0.86 CHRNA7 (0.42) ALDH1A1HPGDESR1ESRRGESR2
SCHEMBL7243631 0.86 CHRNA7 (0.42) ALDH1A1HPGDESR1ESRRGESR2
SCHEMBL7224860 0.86 KDM4E (0.55) KDM4ESMN1; SMN2NPC1ALDH1A1GLA
SCHEMBL7243634 0.86 CHRNA7 (0.42) ALDH1A1HPGDESR1ESRRGESR2
SCHEMBL7231998 0.84 CHRNB2 (0.35) CTSCNPC1MAPTLMNA
SCHEMBL7232602 0.83 CHRNA7 (0.38) CTSCCHRNA7HTR3EHTR3BHTR3A
SCHEMBL7223423 0.83 SLC6A2 (0.35) CTSCMAPTLMNA
SCHEMBL7224906 0.82 CHRNA7 (0.38) KDM4ESMN1; SMN2NPC1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed