SCHEMBL7227965

SCHEMBL7227965

CCN1CCC(N2CC(COS(C)(=O)=O)OC2=O)CC1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 3/20 0.37
CCR5 P51681 2/20 0.35
ADRB3 P13945 1/20 0.34
PARP2 Q9UGN5 1/20 0.32
CCR8 P51685 6/20 0.32
MAOA P21397 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7313802 0.87 HTR2B (0.36) HTR2BCCR5ADRB3MAOA
SCHEMBL12356915 0.84 HTR2B (0.40) HTR2BADRB3CCR8MAOA
SCHEMBL12356916 0.84 HTR2B (0.40) HTR2BADRB3CCR8MAOA
SCHEMBL7229332 0.84 HTR2B (0.38) HTR2BCCR5ADRB3PARP2MAOA
SCHEMBL7310189 0.83 RECQL (0.48) HTR2BCCR8
SCHEMBL7307020 0.81 MAPK1 (0.35)
SCHEMBL7306591 0.78 TP53 (0.42)
SCHEMBL7316915 0.76 MAPK1 (0.45)
SCHEMBL8655209 0.74 HTR2B (0.36) HTR2B
SCHEMBL8858116 0.74 KDM4E (0.35) HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602876-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2003-08-05 US disclosed
US-6204280-B1 OXAZOLIDINONE DERIVATIVE, ANTICOAGULANT MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 2001-03-20 US disclosed
EP-0710657-B1 Antagonists of adhesion receptors MERCK PATENT GMBH (DE) 1998-08-26 EP disclosed
EP-0710657-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-08 EP disclosed