SCHEMBL7229332

SCHEMBL7229332

CC(C)N1CCC(N2CC(COS(C)(=O)=O)OC2=O)CC1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 3/20 0.38
HRH3 Q9Y5N1 3/20 0.33
ADRB3 P13945 1/20 0.33
CCR5 P51681 1/20 0.32
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
MAOA P21397 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7313802 0.86 HTR2B (0.36) HTR2BADRB3CCR5MAOA
SCHEMBL7227965 0.84 HTR2B (0.37) HTR2BADRB3CCR5PARP2MAOA
SCHEMBL12356915 0.83 HTR2B (0.40) HTR2BADRB3MAOA
SCHEMBL12356916 0.83 HTR2B (0.40) HTR2BADRB3MAOA
SCHEMBL8858105 0.81 HTR2B (0.40) HTR2B
SCHEMBL7306687 0.79 MAPK1 (0.35) HRH3
SCHEMBL8858102 0.79 L3MBTL1 (0.38) HTR2B
SCHEMBL7310189 0.78 RECQL (0.48) HTR2B
SCHEMBL7306591 0.78 TP53 (0.42)
SCHEMBL8659488 0.76 HTR2B (0.37) HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602876-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2003-08-05 US disclosed
US-6204280-B1 OXAZOLIDINONE DERIVATIVE, ANTICOAGULANT MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 2001-03-20 US disclosed
EP-0710657-B1 Antagonists of adhesion receptors MERCK PATENT GMBH (DE) 1998-08-26 EP disclosed
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed
EP-0710657-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-08 EP disclosed