SCHEMBL7229145

SCHEMBL7229145

COC(=O)C(Cc1ccc(OCC2CN(CC3CCN(C)CC3)C(=O)O2)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
YAP1 P46937 5/20 0.46
SCN9A Q15858 7/20 0.41
HRH2 P25021 1/20 0.40
HRH1 P35367 1/20 0.40
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
CACNA1B Q00975 2/20 0.39
SRC P12931 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7231433 0.93 ITGB3 (0.47) YAP1SCN9AHRH2HRH1ITGB3
SCHEMBL7237796 0.84 MAPK1 (0.41) YAP1
SCHEMBL7228364 0.83 YAP1 (0.48) YAP1HRH2HRH1CACNA1B
SCHEMBL7229032 0.82 HRH2 (0.47) YAP1HRH2HRH1ITGB3ITGA2B
SCHEMBL7237702 0.82 HRH2 (0.47) YAP1HRH2HRH1ITGB3ITGA2B
SCHEMBL7235737 0.81 ITGB3 (0.45) YAP1ITGB3ITGA2B
SCHEMBL7228437 0.80 YAP1 (0.42) YAP1SCN9AHRH2HRH1ITGB3
SCHEMBL7229147 0.80 MAPK1 (0.38)
SCHEMBL7230827 0.79 MAPK1 (0.39) YAP1HRH2HRH1ITGB3ITGA2B
SCHEMBL7231437 0.79 MAPK1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602876-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2003-08-05 US disclosed
US-6204280-B1 OXAZOLIDINONE DERIVATIVE, ANTICOAGULANT MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 2001-03-20 US disclosed
EP-0710657-B1 Antagonists of adhesion receptors MERCK PATENT GMBH (DE) 1998-08-26 EP disclosed
EP-0710657-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-08 EP disclosed