SCHEMBL7230387

SCHEMBL7230387

COc1cncc(C2(C#N)CC3CCC(C2)N3C)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.40
CYP11B1 P15538 3/20 0.35
CYP11B2 P19099 3/20 0.35
OPRL1 P41146 1/20 0.34
CHRNB2 P17787 6/20 0.33
CHRNA4 P43681 6/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.33
BACE1 P56817 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32
CHRNB4 P30926 5/20 0.32
CHRNA3 P32297 5/20 0.32
CYP1A2 P05177 1/20 0.32
CHRNA7 P36544 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7221029 0.86 CHRNB2 (0.36) CYP11B1CYP11B2OPRL1CHRNB2CHRNA4
SCHEMBL7971885 0.85 KMT2A (0.34) KMT2ACYP11B1CYP11B2OPRL1CHRNB2
SCHEMBL16139986 0.83 OPRL1 (0.36) OPRL1CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL7227978 0.83 CHRNB2 (0.34) CYP11B1CYP11B2OPRL1CHRNB2CHRNA4
SCHEMBL7223956 0.82 OPRL1 (0.36) CYP11B1CYP11B2OPRL1BACE1BACE2
SCHEMBL7223397 0.82 OPRL1 (0.36) CYP11B2OPRL1
SCHEMBL6617335 0.82 OPRL1 (0.41) CYP11B1CYP11B2OPRL1CHRNB2CHRNA4
SCHEMBL7222900 0.82 OPRL1 (0.36) OPRL1CHRNB2CHRNA4
SCHEMBL7223737 0.82 OPRL1 (0.36) CYP11B2OPRL1CHRNB2CHRNA4KDM4E
SCHEMBL7228554 0.82 CHRNB2 (0.43) OPRL1CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6573275-B1 Insecticidal compositions comprising and to methods of combatting and controlling insect pests therewith. SYNGENTA LIMITED (GB) 2003-06-03 US disclosed
EP-0828739-B1 BICYCLIC AMINES AS INSECTICIDES SYNGENTA LTD (GB) 2002-09-11 EP disclosed
US-6207676-B1 Bicyclic amines ZENECA LIMITED (GB) 2001-03-27 US disclosed