SCHEMBL7230402

SCHEMBL7230402

Cc1ccc(Sc2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)nc1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
HTR1A P08908 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7233041 0.89 SLC6A4 (0.34) SLC6A4SLC6A3ALDH1A1HPGD
SCHEMBL7232569 0.88 NPC1 (0.34) SLC6A2SLC6A4SLC6A3NPC1RAB9A
SCHEMBL7232207 0.85 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3NPC1RAB9A
SCHEMBL7224430 0.84 CHRNA7 (0.40) NPC1RAB9AALDH1A1HPGD
SCHEMBL7224129 0.84 NPC1 (0.32) SLC6A2SLC6A4SLC6A3NPC1RAB9A
SCHEMBL7225000 0.83 NPC1 (0.34) SLC6A2SLC6A4SLC6A3NPC1RAB9A
SCHEMBL7232219 0.83 SLC6A3 (0.35) SLC6A2SLC6A4SLC6A3NPC1RAB9A
SCHEMBL7231162 0.83 NPC1 (0.43) SLC6A2SLC6A4SLC6A3NPC1RAB9A
SCHEMBL7223147 0.82 HDAC1 (0.41) SLC6A2SLC6A4SLC6A3NPC1RAB9A
SCHEMBL7230649 0.82 NPC1 (0.32) SLC6A2SLC6A4SLC6A3NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed