SCHEMBL7230653

SCHEMBL7230653

[CH]CCC(C)NC(=O)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.41
KCNH2 Q12809 1/20 0.41
MLYCD O95822 4/20 0.36
CA2 P00918 2/20 0.34
ALDH1A1 P00352 2/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
EPHX1 P07099 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
TAS1R2 Q8TE23 1/20 0.31
HPGD P15428 1/20 0.31
CA3 P07451 2/20 0.31
CA5A P35218 2/20 0.31
CA5B Q9Y2D0 2/20 0.31
CA12 O43570 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL995905 0.82 MLYCD (0.43) ESR1KCNH2MLYCDCA2ALDH1A1
SCHEMBL7230655 0.82 ALDH1A1 (0.46) ESR1KCNH2MLYCDCA2ALDH1A1
SCHEMBL566464 0.78 MLYCD (0.41) ESR1KCNH2MLYCDCA2ALDH1A1
SCHEMBL566465 0.78 MLYCD (0.41) ESR1KCNH2MLYCDCA2ALDH1A1
SCHEMBL7045874 0.77 MLYCD (0.57) ESR1KCNH2MLYCDMEN1KMT2A
SCHEMBL8060275 0.77 ESR1 (0.44) ESR1KCNH2MLYCDCA2ALDH1A1
SCHEMBL31496034 0.77 ESR1 (0.44) ESR1KCNH2MLYCDCA2ALDH1A1
SCHEMBL9344459 0.77 SMN1; SMN2 (0.47) ESR1KCNH2MLYCDCA2ALDH1A1
SCHEMBL8060272 0.77 ESR1 (0.44) ESR1KCNH2MLYCDCA2ALDH1A1
SCHEMBL12926140 0.76 MLYCD (0.39) ESR1KCNH2MLYCDCA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6534503-B1 Treating sexual dysfunction, such as erectile dysfunction or sexual arousal disorder, with a compound having the generic formula X1-X2-(D)Phe-Arg-(D)Trp-X3. A particularly useful compound is HP-228, which has the formula LION BIOSCIENCE AG (DE) 2003-03-18 US claimed
EP-1214330-A1 BENZIMIDAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-06-19 EP claimed
WO-2001021634-A1 BENZIMIDAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-03-29 WO claimed
EP-1214330-A1 BENZIMIDAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-06-19 EP disclosed
WO-2001021634-A1 BENZIMIDAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-03-29 WO disclosed