SCHEMBL7230723

SCHEMBL7230723

CC(C)(C)OC(=O)NC(=N)C(CN1CCNCC1)N1CC(COc2ccc(CC(NC(=O)OC(C)(C)C)C(=O)O)cc2)OC1=O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.42
ITGA2B P08514 10/20 0.42
PTPN1 P18031 3/20 0.40
YAP1 P46937 1/20 0.37
ITGAV P06756 1/20 0.37
HRH2 P25021 1/20 0.36
HRH1 P35367 1/20 0.36
MAPK1 P28482 1/20 0.36
ITGA4 P13612 1/20 0.35
ITGB7 P26010 1/20 0.35
ACE P12821 1/20 0.35
HDAC8 Q9BY41 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7230083 0.94 ITGB3 (0.44) ITGB3ITGA2BPTPN1YAP1ITGAV
SCHEMBL7237897 0.94 YAP1 (0.37) ITGB3ITGA2BPTPN1YAP1HRH2
SCHEMBL7237989 0.93 ITGB3 (0.46) ITGB3ITGA2BPTPN1ITGAVHRH2
SCHEMBL7229494 0.89 ITGB3 (0.48) ITGB3ITGA2BITGAV
SCHEMBL7237720 0.89 ITGB3 (0.44) ITGB3ITGA2BPTPN1YAP1ITGAV
SCHEMBL7229611 0.89 ITGB3 (0.46) ITGB3ITGA2BPTPN1YAP1ITGAV
SCHEMBL7229317 0.88 ITGB3 (0.39) ITGB3ITGA2BPTPN1YAP1HRH2
SCHEMBL7227732 0.88 ITGB3 (0.48) ITGB3ITGA2BPTPN1ITGAV
SCHEMBL7228009 0.87 ITGB3 (0.41) ITGB3ITGA2BYAP1HRH2HRH1
SCHEMBL7238373 0.86 ITGB3 (0.43) ITGB3ITGA2BPTPN1YAP1ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602876-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2003-08-05 US disclosed
US-6204280-B1 OXAZOLIDINONE DERIVATIVE, ANTICOAGULANT MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 2001-03-20 US disclosed
EP-0710657-B1 Antagonists of adhesion receptors MERCK PATENT GMBH (DE) 1998-08-26 EP disclosed
EP-0710657-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-08 EP disclosed