SCHEMBL7230828

SCHEMBL7230828

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ncc(-c2ccc(Cl)c(Cl)c2)o1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 4/20 0.41
SLC6A4 P31645 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
ITGA5 P08648 1/20 0.36
CHRNB1 P11230 1/20 0.36
CHRNB2 P17787 1/20 0.36
SLC6A2 P23975 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
CHRND Q07001 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7231985 0.89 HDAC1 (0.46) SLC6A3SLC6A4CA12CA1CA2
SCHEMBL7232162 0.87 HDAC1 (0.50) CA12CA1CA2CA4NPC1
SCHEMBL7231176 0.87 CA12 (0.39) SLC6A3SLC6A4CA12CA1CA2
SCHEMBL7233445 0.86 CA12 (0.41) CA12CA1CA2CA4CHRNB2
SCHEMBL7226687 0.85 TUBB4A (0.46) CA12CA1CA2CA4NPC1
SCHEMBL7226619 0.85 HDAC1 (0.46) SLC6A3CA12CA1CA2CA4
SCHEMBL7222561 0.85 CA12 (0.48) CA12CA1CA2CA4CHRNB2
SCHEMBL7234526 0.85 HDAC1 (0.47) SLC6A3CA12CA1CA2CA4
SCHEMBL7224305 0.85 HDAC1 (0.46) SLC6A3SLC6A4CA12CA1CA2
SCHEMBL7073214 0.84 TUBB4A (0.47) CA12CA1CA2CA4CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed