SCHEMBL7230944

SCHEMBL7230944

COc1cc(-c2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)ccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
CTSC P53634 1/20 0.40
TEC P42680 1/20 0.39
TXK P42681 1/20 0.39
BTK Q06187 1/20 0.39
ITK Q08881 1/20 0.39
CHRNA7 P36544 8/20 0.37
HTR3E A5X5Y0 4/20 0.37
HTR3B O95264 4/20 0.37
HTR3A P46098 4/20 0.37
HTR3D Q70Z44 4/20 0.37
HTR3C Q8WXA8 4/20 0.37
EGLN1 Q9GZT9 2/20 0.36
USP30 Q70CQ3 1/20 0.36
HPGDS O60760 1/20 0.36
MAPK13 O15264 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7230436 0.87 CTSS (0.42) CTSSCTSKTECTXKBTK
SCHEMBL7224866 0.87 CTSC (0.40) CTSCTECTXKBTKITK
SCHEMBL7224824 0.85 CHRNA7 (0.38) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7223916 0.84 CTSC (0.35) CTSSCTSKCTSCEGLN1
SCHEMBL7232573 0.83 CTSC (0.34) CTSCEGLN1
SCHEMBL7224193 0.83 HDAC3 (0.53) CTSSCTSKCHRNA7HTR3EHTR3B
SCHEMBL7232229 0.83 HDAC6 (0.50) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7224860 0.82 KDM4E (0.55) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7226599 0.82 KDM4E (0.37) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7233013 0.81 RXFP1 (0.47) CHRNA7HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed