SCHEMBL7230962

SCHEMBL7230962

COc1ccc2c(c1)-c1nc(Nc3cccc(OCc4ccccc4)c3)ncc1CC2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.56
FYN P06241 1/20 0.55
CDK2 P24941 4/20 0.53
CCNA2 P20248 3/20 0.53
CDK5 Q00535 1/20 0.53
CDK5R1 Q15078 1/20 0.53
PLK1 P53350 3/20 0.49
AURKA O14965 1/20 0.49
CCNA1 P78396 1/20 0.49
IKBKB O14920 1/20 0.49
CDK1 P06493 1/20 0.49
IGF1R P08069 4/20 0.49
MEN1 O00255 1/20 0.47
USP2 O75604 1/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CASP1 P29466 1/20 0.47
CYP2C19 P33261 1/20 0.47
CASP7 P55210 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17560321 0.90 KDR (0.64) KDRFYNCDK2CCNA2CDK5
SCHEMBL7232833 0.86 KDR (0.55) KDRFYNCDK2CCNA2IKBKB
SCHEMBL6999967 0.84 KDR (0.65) KDRFYNCDK2CCNA2CDK5
SCHEMBL7230996 0.83 FYN (0.68) KDRFYNCDK2CCNA2CDK5
SCHEMBL7241504 0.82 FYN (0.58) KDRFYNCDK2CCNA2CDK5
SCHEMBL7238444 0.82 FYN (0.58) KDRFYNCDK2CCNA2CDK5
SCHEMBL6996576 0.82 IGF1R (0.55) KDRFYNCDK2CCNA2CDK5
SCHEMBL7001192 0.80 SYK (0.54) KDRFYNCDK2CCNA2CDK5
SCHEMBL7241524 0.79 CDK2 (0.59) KDRFYNCDK2CCNA2CDK5
SCHEMBL6994864 0.79 KDR (0.63) KDRFYNCDK2CCNA2CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6599908-B1 Potent and selective inhibitors of the protein tyrosine kinases p56lck and p59fyn CELLTECH R & D LIMITED (GB) 2003-07-29 US disclosed
US-6057329-A Fused polycyclic 2-aminopyrimidine derivatives CELLTECH THERAPEUTICS LIMITED (GB) 2000-05-02 US disclosed