SCHEMBL7232602

SCHEMBL7232602

COc1ncc(-c2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)s1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 9/20 0.38
HTR3E A5X5Y0 5/20 0.35
HTR3B O95264 5/20 0.35
HTR3A P46098 5/20 0.35
HTR3D Q70Z44 5/20 0.35
HTR3C Q8WXA8 5/20 0.35
SLC6A3 Q01959 1/20 0.35
CTSC P53634 1/20 0.35
AKT1 P31749 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7232814 0.87 CHRNA7 (0.37) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7231089 0.85 CHRNA7 (0.37) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7231604 0.84 SLC6A3 (0.32) SLC6A3
SCHEMBL7225345 0.84 CHRNA7 (0.41) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7233001 0.84 CHRNA7 (0.38) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7232991 0.83 SLC6A3 (0.32) SLC6A3
SCHEMBL7225220 0.83 CHRNA7 (0.39) CHRNA7
SCHEMBL7224906 0.83 CHRNA7 (0.38) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7224866 0.83 CTSC (0.40) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7224299 0.83 NPC1 (0.45) CHRNA7HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed