SCHEMBL7233182

SCHEMBL7233182

COC(=O)CCc1c(-c2ccc(C(F)(F)F)cc2)[nH]c2ccc(Cl)cc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.50
TSPO P30536 1/20 0.48
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
HPGD P15428 1/20 0.45
CYP2C19 P33261 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HSD17B10 Q99714 1/20 0.45
CYP2C9 P11712 1/20 0.43
EGFR P00533 2/20 0.42
SRC P12931 1/20 0.42
TUBB4A P04350 2/20 0.42
TUBB P07437 2/20 0.42
TUBA3C P0DPH7 2/20 0.42
TUBA1B P68363 2/20 0.42
TUBA4A P68366 2/20 0.42
TUBB4B P68371 2/20 0.42
TUBB3 Q13509 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7236310 0.94 TACR1 (0.49) TACR1TSPOKDM4EALDH1A1CYP1A2
SCHEMBL7798973 0.94 TACR1 (0.48) TACR1TSPOKDM4EALDH1A1CYP1A2
SCHEMBL7242930 0.87 PPARG (0.50) TACR1TSPOKDM4EALDH1A1CYP1A2
SCHEMBL22160195 0.86 TACR1 (0.51) TACR1CYP2C9EGFRSRC
SCHEMBL7238513 0.84 TSPO (0.56) TACR1TSPOKDM4EALDH1A1CYP1A2
SCHEMBL7233540 0.83 TSPO (0.47) TACR1TSPOKDM4EALDH1A1CYP1A2
SCHEMBL7241810 0.82 CXCR2 (0.56) TACR1TSPOCYP2C9
SCHEMBL7790369 0.82 CXCR2 (0.52) TACR1TSPOKDM4EALDH1A1CYP1A2
SCHEMBL7232797 0.81 TACR1 (0.43) TACR1TSPOKDM4EALDH1A1CYP1A2
SCHEMBL7238595 0.80 CXCR2 (0.53) TACR1TSPOKDM4EALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6605633-B1 Such as 5-Bromo-2-phenyl-1H-indole-3-butanoic acid FOURNIER INDUSTRIE ET SANTE (FR) 2003-08-12 US disclosed