SCHEMBL7233242

SCHEMBL7233242

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(-c2ncc(Cl)o2)s1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 5/20 0.36
CHRNA7 P36544 12/20 0.36
HTR3E A5X5Y0 5/20 0.34
HTR3B O95264 5/20 0.34
HTR3A P46098 5/20 0.34
HTR3D Q70Z44 5/20 0.34
HTR3C Q8WXA8 5/20 0.34
CHRNB2 P17787 5/20 0.33
CHRNA4 P43681 5/20 0.33
CHRNB4 P30926 2/20 0.33
CHRNA3 P32297 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CHRNA1 P02708 1/20 0.33
CHRNG P07510 1/20 0.33
CHRNB1 P11230 1/20 0.33
HPGD P15428 1/20 0.33
CHRND Q07001 1/20 0.33
CHRNA2 Q15822 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7225477 0.88 CHRNA7 (0.36) AKT1CHRNA7HTR3EHTR3BHTR3A
SCHEMBL7232339 0.85 CHRNA7 (0.36) AKT1CHRNA7HTR3EHTR3BHTR3A
SCHEMBL7231059 0.85 ALDH1A1 (0.38) AKT1CHRNA7HTR3EHTR3BHTR3A
SCHEMBL7230457 0.85 CHRNA7 (0.37) AKT1CHRNA7HTR3EHTR3BHTR3A
SCHEMBL7231089 0.85 CHRNA7 (0.37) AKT1CHRNA7HTR3EHTR3BHTR3A
SCHEMBL7225620 0.84 AKT1 (0.37) AKT1CHRNA7HTR3EHTR3BHTR3A
SCHEMBL7223964 0.82 CHRNA7 (0.42) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7243634 0.82 CHRNA7 (0.42) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7243631 0.82 CHRNA7 (0.42) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7224923 0.82 AKT1 (0.36) AKT1CHRNA7HTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed