SCHEMBL7240669

SCHEMBL7240669

COC(=O)CCc1ccc(C(=O)NC[C@H](NC(=O)OCc2ccccc2)C(=O)O)s1

nearest known ligand 0.74

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 15/20 0.74
ITGAV P06756 15/20 0.74
ITGA2B P08514 7/20 0.74
CASP1 P29466 1/20 0.45
KYNU Q16719 1/20 0.43
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.42
SIRT1 Q96EB6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016434 0.90 ITGB3 (0.61) ITGB3ITGAVITGA2BCASP1KYNU
SCHEMBL6016218 0.85 ITGB3 (0.75) ITGB3ITGAVITGA2BCASP1
SCHEMBL6016219 0.83 ITGB3 (0.60) ITGB3ITGAVITGA2BCASP1CTSL
SCHEMBL3370106 0.82 CASP1 (0.53) ITGB3ITGAVITGA2BCASP1KYNU
SCHEMBL5626356 0.81 ITGB3 (0.63) ITGB3ITGAVITGA2BKYNUCTSL
SCHEMBL5626363 0.81 ITGB3 (0.63) ITGB3ITGAVITGA2BKYNUCTSL
SCHEMBL6016166 0.79 ITGB3 (1.00) ITGB3ITGAVITGA2B
SCHEMBL6016256 0.78 ITGB3 (0.62) ITGB3ITGAVITGA2BCASP1CTSL
SCHEMBL7370216 0.76 CTSK (0.57) ITGB3ITGAVKYNUCTSLCTSB
SCHEMBL7370220 0.76 CTSK (0.57) ITGB3ITGAVKYNUCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6566366-B1 For therapy of tumor growth, osteoporosis, inflammation and cardiovascular disorders AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-05-20 US disclosed