SCHEMBL7243745

SCHEMBL7243745

CC(C)(C)OC(=O)N(Cc1cc(NC(=N)N[N+](=O)[O-])cc(C(F)(F)F)c1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CETP P11597 4/20 0.38
P2RX1 P51575 4/20 0.35
MAPT P10636 2/20 0.34
CACNA1G O43497 1/20 0.34
CACNA1B Q00975 1/20 0.34
CACNA1C Q13936 1/20 0.34
TMPRSS4 Q9NRS4 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 2/20 0.32
BMP1 P13497 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
RAF1 P04049 1/20 0.32
BRAF P15056 1/20 0.32
TACR1 P25103 2/20 0.32
GPR35 Q9HC97 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7243748 0.82 CETP (0.36) CETPP2RX1MAPTCACNA1GCACNA1B
SCHEMBL6676867 0.80 CETP (0.40) CETPMAPTCACNA1GCACNA1BCACNA1C
SCHEMBL6677408 0.78 CETP (0.42) CETPP2RX1CACNA1GCACNA1BCACNA1C
SCHEMBL6674825 0.78 P2RX1 (0.39) P2RX1MAPTTMPRSS4LMNAMEN1
Hydrochloric Acid SCHEMBL6681155 0.77 P2RX1 (0.38) P2RX1MAPTTMPRSS4LMNAMEN1
SCHEMBL7240779 0.75 NR1H4 (0.35) ALDH1A1LMNA
SCHEMBL6678261 0.73 CETP (0.43) CETPCACNA1GCACNA1BCACNA1CTACR1
SCHEMBL6681975 0.71 AKT1 (0.44)
SCHEMBL6690431 0.68 BACE1 (0.41) MAPTMEN1KMT2A
SCHEMBL10384367 0.68 MAPT (0.52) MAPTALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed