SCHEMBL7243748

SCHEMBL7243748

CC(C)(C)OC(=O)N(Cc1cc(NC(N)=N[N+](=O)[O-])cc(C(F)(F)F)c1)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CETP P11597 3/20 0.36
CACNA1G O43497 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNA1C Q13936 1/20 0.35
SIGMAR1 Q99720 3/20 0.34
P2RX1 P51575 4/20 0.34
GRM2 Q14416 1/20 0.34
RAF1 P04049 1/20 0.33
BRAF P15056 1/20 0.33
MAPT P10636 2/20 0.33
TMPRSS4 Q9NRS4 1/20 0.32
ALDH1A1 P00352 2/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6684630 0.86 GPR35 (0.37) SIGMAR1P2RX1MAPTTMPRSS4ALDH1A1
SCHEMBL6676867 0.82 CETP (0.40) CETPCACNA1GCACNA1BCACNA1CGRM2
SCHEMBL7243745 0.82 CETP (0.38) CETPCACNA1GCACNA1BCACNA1CP2RX1
SCHEMBL6674828 0.79 SIGMAR1 (0.39) SIGMAR1P2RX1RAF1BRAFMAPT
Hydrochloric Acid SCHEMBL6681157 0.78 SIGMAR1 (0.40) SIGMAR1P2RX1RAF1BRAFMAPT
SCHEMBL6677408 0.77 CETP (0.42) CETPCACNA1GCACNA1BCACNA1CP2RX1
SCHEMBL7240782 0.75 MAPT (0.32) GRM2MAPTALDH1A1
SCHEMBL6678261 0.74 CETP (0.43) CETPCACNA1GCACNA1BCACNA1CGRM2
SCHEMBL6681977 0.71 AKT1 (0.43) SIGMAR1
SCHEMBL6690435 0.68 NOS3 (0.53) SIGMAR1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed