SCHEMBL7243797

SCHEMBL7243797

CCn1c(CCOC)cc2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.39
GRIK1 P39086 1/20 0.38
GRIK2 Q13002 1/20 0.38
AGTR1 P30556 1/20 0.37
AGTR2 P50052 1/20 0.37
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.37
USP2 O75604 1/20 0.37
GLA P06280 1/20 0.37
TSHR P16473 1/20 0.37
ALOX12 P18054 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
MTNR1A P48039 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11603605 0.80 PPARG (0.45) PPARGAGTR1AGTR2TSHRCA12
SCHEMBL7246243 0.80 NPC1 (0.49) KMT2ARAB9ANPC1
SCHEMBL11375360 0.80 PPARG (0.40) PPARGAGTR1AGTR2KMT2AALDH1A1
SCHEMBL11504340 0.79 HTT (0.42) PPARGKMT2AALDH1A1MEN1USP2
SCHEMBL7243803 0.77 HPGD (0.46) KMT2AALDH1A1GLATSHRCASP7
SCHEMBL11390081 0.76 CA12 (0.43) PPARGAGTR1AGTR2KMT2AALDH1A1
SCHEMBL28206798 0.76 CA12 (0.40) PPARGKMT2AALDH1A1MEN1USP2
SCHEMBL11389628 0.76 HTT (0.43) KMT2AALDH1A1MEN1USP2TSHR
SCHEMBL11396410 0.76 CA12 (0.40) PPARGAGTR1AGTR2KMT2AALDH1A1
SCHEMBL13307121 0.75 ALDH1A1 (0.45) KMT2AALDH1A1MEN1TSHRMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6503907-B2 Indole derivatives or dihydroindole derivatives or salts are useful for the treatment of diseases associated with 2,3-oxidosqualene-lanosterol cyclase such as gallstone, tumorhypercholesterolemia, hyperlipemia, arterioscerosis etc. HOFFMANN-LA ROCHE INC. 2003-01-07 US disclosed