SCHEMBL7244459

SCHEMBL7244459

CS(=O)(=O)N(Cc1ccccc1)c1cccc([C@H](O)CN(CCOc2ccc3c(c2)[nH]c2ccccc23)Cc2ccccc2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 2/20 0.40
CTSV O60911 1/20 0.38
CTSL P07711 1/20 0.38
MAOB P27338 2/20 0.36
HCRTR2 O43614 2/20 0.35
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PER2 O15055 2/20 0.35
MAOA P21397 1/20 0.35
CRY1 Q16526 1/20 0.35
CRY2 Q49AN0 1/20 0.35
GRM2 Q14416 1/20 0.35
ALK Q9UM73 1/20 0.34
ADRB3 P13945 1/20 0.34
ADRA1A P35348 1/20 0.34
ATM Q13315 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7526000 1.00 NR1H3 (0.40) NR1H3CTSVCTSLMAOBHCRTR2
SCHEMBL7248052 1.00 NR1H3 (0.40) NR1H3CTSVCTSLMAOBHCRTR2
SCHEMBL5194303 0.90 NR1H3 (0.38) NR1H3MAOBHCRTR2ACHEMEN1
SCHEMBL5193993 0.89 NR1H3 (0.37) NR1H3MAOBHCRTR2ACHEMEN1
SCHEMBL7250840 0.87 ATM (0.40) NR1H3CTSVCTSLMAOBHCRTR2
SCHEMBL1120784 0.87 NPSR1 (0.39) NR1H3MAOBACHEMAOAALK
Hydrochloric Acid SCHEMBL7616039 0.85 ADRB3 (0.48) ADRB3ADRA1A
SCHEMBL6746794 0.84 NR1H3 (0.41) NR1H3CTSVCTSLMAOBHCRTR2
SCHEMBL6744765 0.84 NR1H3 (0.41) NR1H3CTSVCTSLMAOBHCRTR2
SCHEMBL7252170 0.83 HCRTR2 (0.41) CTSVCTSLMAOBHCRTR2BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6599892-B2 Beta-lactamase inhitiors RESEARCH CORPORATION TECHNOLOGIES, INC. 2003-07-29 US disclosed
US-20030045727-A1 Process for preparing optically active secondary alcohols having nitrogenous or oxygenic functional groups ASAHI KASEI KABUSHIKI KAISHA (JP) 2003-03-06 US disclosed
EP-1254885-A1 PROCESS FOR PREPARING OPTICALLY ACTIVE SECONDARY ALCOHOLS HAVING NITROGENOUS OR OXYGENIC FUNCTIONAL GROUPS Asahi Kasei Kabushiki Kaisha (JP) 2002-11-06 EP disclosed
US-20020025954-A1 7-alkylidene cephalosporanic acid derivatives and methods of using the same RESEARCH CORPORATION TECHNOLOGIES, INC. 2002-02-28 US disclosed
US-6303592-B1 AS INHIBITORS OF .BETA.-LACTAMASE ENZYMES RESEARCH CORPORATION TECHNOLOGIES, INC. 2001-10-16 US disclosed
WO-1996017849-A1 7-ALKYLIDENE CEPHALOSPORANIC ACID DERIVATIVES AND METHODS OF USING THE SAME RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1996-06-13 WO disclosed
WO-1996017848-A1 7-VINYLIDENE CEPHALOSPORINS AND METHODS OF USING THE SAME SOUTHERN METHODIST UNIVERSITY (US) 1996-06-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030045727-A1 Process for preparing optically active secondary alcohols having nitrogenous or oxygenic functional groups ADH1A, ADH5, ADH1C NR1H3 53/4885CTSV 4705/4885CTSL 4734/4885
US-20020025954-A1 7-alkylidene cephalosporanic acid derivatives and methods of using the same STS, PEPD, IDUA NR1H3 3232/4885CTSV 728/4885CTSL 343/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.