SCHEMBL7249651

SCHEMBL7249651

[CH2]c1nc2ccncc2[nH]1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.50
ALDH1A1 P00352 5/20 0.50
RAB9A P51151 5/20 0.50
PKM P14618 4/20 0.50
NPC1 O15118 4/20 0.50
KDM4E B2RXH2 4/20 0.50
HPGD P15428 2/20 0.50
METAP1 P53582 2/20 0.49
METAP2 P50579 1/20 0.49
ADORA3 P0DMS8 1/20 0.46
AURKA O14965 1/20 0.46
RPS6KA5 O75582 1/20 0.45
PDE5A O76074 2/20 0.44
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
HPSE Q9Y251 1/20 0.43
KRAS P01116 1/20 0.41
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1170780 0.78 ALDH1A1 (0.68) SMN1; SMN2ALDH1A1RAB9APKMNPC1
SCHEMBL879284 0.75 ALDH1A1 (0.50) SMN1; SMN2ALDH1A1RAB9APKMNPC1
SCHEMBL21496798 0.75 ALDH1A1 (0.50) SMN1; SMN2ALDH1A1RAB9APKMNPC1
SCHEMBL15088513 0.75 SMN1; SMN2 (0.50) SMN1; SMN2ALDH1A1RAB9APKMNPC1
SCHEMBL34462940 0.75 SMN1; SMN2 (0.50) SMN1; SMN2ALDH1A1RAB9APKMNPC1
SCHEMBL9698797 0.75 ALDH1A1 (0.55) SMN1; SMN2ALDH1A1RAB9APKMNPC1
SCHEMBL2106050 0.75 SMN1; SMN2 (0.50) SMN1; SMN2ALDH1A1RAB9APKMNPC1
SCHEMBL18757848 0.73 RAB9A (0.56) SMN1; SMN2ALDH1A1RAB9APKMNPC1
SCHEMBL5398 0.71 ALDH1A1 (0.60) SMN1; SMN2ALDH1A1RAB9APKMNPC1
SCHEMBL23771281 0.71 RAB9A (0.57) SMN1; SMN2ALDH1A1RAB9APKMNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6610731-B2 Antiinflammatory BRISTOL-MYERS SQUIBB COMPANY 2003-08-26 US disclosed
US-6403632-B1 CYCLIC AMIDE DERIVATIVE BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-06-11 US disclosed