SCHEMBL7250216

SCHEMBL7250216

COc1ccccc1Oc1c(Cl)nc(-c2cc[n+]([O-])cc2)nc1NS(=O)(=O)c1ncc(C)s1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 14/20 0.46
EDNRB P24530 9/20 0.46
DHPS P49366 6/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7248679 0.91 EDNRA (0.57) EDNRAEDNRBDHPS
SCHEMBL6972015 0.84 DHPS (0.53) EDNRAEDNRBDHPS
SCHEMBL6969386 0.84 EDNRA (0.53) EDNRAEDNRBDHPS
SCHEMBL5035301 0.84 EDNRA (0.66) EDNRAEDNRB
SCHEMBL6957003 0.83 EDNRA (0.47) EDNRAEDNRBDHPS
SCHEMBL6972208 0.83 DHPS (0.53) EDNRAEDNRBDHPS
SCHEMBL6972565 0.81 EDNRA (0.47) EDNRAEDNRBDHPS
SCHEMBL5032747 0.81 EDNRA (0.67) EDNRAEDNRB
SCHEMBL6961198 0.80 EDNRA (0.47) EDNRAEDNRBDHPS
SCHEMBL6959001 0.80 EDNRA (0.62) EDNRAEDNRBDHPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6521631-B2 N-(6-methoxy-5-(2-methoxy-phenoxy)-2-pyridin-4-yl-pyrimidin-4 -yl)) 5-isopropyl-pyridine-2-sulfonamide; treatment of disorders which are associated with abnormal vascular tone and endothelial dysfunction. HOFFMANN-LA ROCHE INC. 2003-02-18 US disclosed