SCHEMBL7250809

SCHEMBL7250809

COC(=O)N1CCN(c2nn(-c3ccc(Cl)cc3)cc2-c2ccncc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.46
MAPT P10636 4/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
GRM5 P41594 1/20 0.44
HIF1A Q16665 2/20 0.44
TRPV1 Q8NER1 1/20 0.43
ALDH1A1 P00352 6/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C19 P33261 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
RAB9A P51151 1/20 0.41
TRPA1 O75762 1/20 0.40
BRAF P15056 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
RGS12 O14924 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7248577 0.82 MAPK14 (0.52) AKR1C3ALDH1A1KMT2ARAB9ADRD2
SCHEMBL5829519 0.79 CYP17A1 (0.51) MAPTHIF1AALDH1A1CYP3A4CYP2C19
SCHEMBL6338216 0.78 GRIA1 (0.47) MAPTSMN1; SMN2GRM5ALDH1A1BRAF
SCHEMBL5829983 0.75 KDM4E (0.41) AKR1C3MAPTSMN1; SMN2GRM5ALDH1A1
SCHEMBL5829985 0.75 KDM4E (0.41) AKR1C3MAPTSMN1; SMN2GRM5ALDH1A1
SCHEMBL5257757 0.74 MAPK11 (0.69) AKR1C3HIF1A
Water SCHEMBL28746870 0.73 MAPK11 (0.68) AKR1C3HIF1A
SCHEMBL14519526 0.72 MAPK11 (0.55) HIF1A
SCHEMBL38663059 0.72 HIF1A (0.76) AKR1C3MAPTSMN1; SMN2HIF1ATRPV1
SCHEMBL6337994 0.70 MELK (0.51) MAPTKMT2AMEN1BRAFDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6617324-B1 Phenyl, cyclohexyl and pyridinyl or pyrimidinyl-substituted G. D. SEARLE & COMPANY 2003-09-09 US disclosed