SCHEMBL7248577

SCHEMBL7248577

CN1CCN(c2nn(-c3ccc(Cl)cc3)cc2-c2ccncc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.52
MAPK11 Q15759 2/20 0.52
MAPK13 O15264 1/20 0.52
MAPK12 P53778 1/20 0.52
MELK Q14680 4/20 0.51
FLT3 P36888 1/20 0.44
GSK3B P49841 1/20 0.44
KMT2A Q03164 1/20 0.42
PTGS2 P35354 1/20 0.41
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
RAB9A P51151 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
ROCK2 O75116 2/20 0.40
ROCK1 Q13464 2/20 0.40
CSNK1D P48730 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6337994 0.87 MELK (0.51) MAPK14MAPK11MAPK13MAPK12MELK
SCHEMBL5829487 0.87 ALDH1A1 (0.51) MAPK14MAPK11MELKKMT2APTGS2
SCHEMBL5829519 0.84 CYP17A1 (0.51) MAPK14MAPK11FLT3GSK3BKMT2A
SCHEMBL7250809 0.82 AKR1C3 (0.46) KMT2AGAARAB9AALDH1A1DRD2
SCHEMBL5829983 0.76 KDM4E (0.41) KMT2ANPC1RAB9AKDM4EALDH1A1
SCHEMBL5829985 0.76 KDM4E (0.41) KMT2ANPC1RAB9AKDM4EALDH1A1
SCHEMBL6310322 0.71 RAB9A (0.50) MAPK14FLT3GSK3BKMT2APTGS2
SCHEMBL8110243 0.70 ALDH1A1 (0.52) MAPK14FLT3GSK3BKMT2APTGS2
SCHEMBL5463406 0.69 ROCK2 (0.44) MAPK14MAPK11MAPK13MAPK12MELK
SCHEMBL28337260 0.69 MELK (0.69) MELKKMT2ANPC1GAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6617324-B1 Phenyl, cyclohexyl and pyridinyl or pyrimidinyl-substituted G. D. SEARLE & COMPANY 2003-09-09 US disclosed