SCHEMBL5829985

SCHEMBL5829985

CCOC(=O)[C@@H]1CN(c2nn(-c3ccc(Cl)cc3)cc2-c2ccncc2)CCN1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
MAPK1 P28482 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
TP53 P04637 3/20 0.41
POLB P06746 2/20 0.41
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
HPGD P15428 3/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP1A2 P05177 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MAPT P10636 4/20 0.37
DRD2 P14416 2/20 0.37
GRM5 P41594 1/20 0.37
USP2 O75604 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5829983 1.00 KDM4E (0.41) KDM4ERAB9ANPC1MAPK1NPSR1
SCHEMBL5456414 0.78 MAPK11 (0.60)
SCHEMBL7248577 0.76 MAPK14 (0.52) KDM4ERAB9ANPC1MAPK1ALDH1A1
SCHEMBL7250809 0.75 AKR1C3 (0.46) RAB9ACYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL5829519 0.71 CYP17A1 (0.51) RAB9ANPC1MAPK1NPSR1CYP3A4
SCHEMBL5452258 0.69 MAPK14 (0.48)
SCHEMBL6310322 0.67 RAB9A (0.50) KDM4ERAB9ANPC1TP53HPGD
SCHEMBL14519748 0.66 MAPK14 (0.48)
SCHEMBL6337994 0.65 MELK (0.51) MEN1KMT2AMAPTDRD2
SCHEMBL11765733 0.65 NPC1 (0.68) KDM4ERAB9ANPC1MAPK1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071198-B1 Antiinflamamtory agents; antiarthritic agents; inflammatory bowel disorders; multiple sclerosis; asthma PHARMACIA CORPORATION (US) 2006-07-04 US disclosed