SCHEMBL7251899

SCHEMBL7251899

NC(=O)c1ccccc1[C@H]1CCCc2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.48
RPS6KB1 P23443 2/20 0.48
AURKB Q96GD4 1/20 0.48
PARP1 P09874 1/20 0.48
PARP2 Q9UGN5 1/20 0.48
HAO1 Q9UJM8 1/20 0.47
ALDH1A1 P00352 2/20 0.47
MAPK1 P28482 1/20 0.46
MAPK14 Q16539 1/20 0.46
CD38 P28907 2/20 0.46
IDO1 P14902 2/20 0.45
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
TAS1R2 Q8TE23 1/20 0.45
ADRA2A P08913 2/20 0.44
ADRA1A P35348 2/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1B P35368 1/20 0.44
HTR1A P08908 1/20 0.44
OPRM1 P35372 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL484230 1.00 AURKA (0.48) AURKARPS6KB1AURKBPARP1PARP2
SCHEMBL3462221 0.90 PIN1 (0.49) AURKARPS6KB1AURKBPARP1PARP2
SCHEMBL3460627 0.90 PIN1 (0.49) AURKARPS6KB1AURKBPARP1PARP2
SCHEMBL2798590 0.90 PIN1 (0.49) AURKARPS6KB1AURKBPARP1PARP2
SCHEMBL15518445 0.86 HAO1 (0.51) HAO1ALDH1A1MAPK1MAPK14TAS1R3
SCHEMBL5272968 0.85 CD38 (0.45) AURKARPS6KB1AURKBPARP1PARP2
Hydrochloric Acid SCHEMBL15520046 0.84 HAO1 (0.50) HAO1ALDH1A1MAPK1MAPK14TAS1R3
SCHEMBL8516651 0.83 AURKA (0.46) AURKARPS6KB1AURKBPARP1PARP2
SCHEMBL14360065 0.79 HAO1 (0.64) HAO1MAPK1MAPK14IDO1ADRA2A
SCHEMBL21001113 0.79 ADRA2A (0.49) AURKARPS6KB1AURKBPARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002094767-A3 TRISUBSTITUTED-N-[(1S)-1,2,3,4-TETRAHYDRO-1-NAPHTHALENYL] BENZAMIDES WHICH INHIBIT P2X3 AND P2X2/3 CONTAINING RECEPTORS ABBOTT LAB (US) 2003-07-31 WO disclosed
WO-2002094767-A2 TRISUBSTITUTED-N-[(1S)-1,2,3,4-TETRAHYDRO-1-NAPHTHALENYL] BENZAMIDES WHICH INHIBIT P2X3 AND P2X2/3 CONTAINING RECEPTORS ABBOTT LABORATORIES (US) 2002-11-28 WO disclosed