SCHEMBL8516651

SCHEMBL8516651

NC(=O)c1cccc(N)c1C1CCCc2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AURKA O14965 3/20 0.46
RPS6KB1 P23443 3/20 0.46
AURKB Q96GD4 1/20 0.46
PARP1 P09874 1/20 0.46
PARP2 Q9UGN5 1/20 0.46
CD38 P28907 2/20 0.43
TAS1R3 Q7RTX0 5/20 0.43
TAS1R1 Q7RTX1 5/20 0.43
TAS1R2 Q8TE23 5/20 0.43
HAO1 Q9UJM8 1/20 0.42
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.41
MAPK14 Q16539 1/20 0.41
PIN1 Q13526 1/20 0.41
GID4 Q8IVV7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8516606 0.92 PIN1 (0.46) AURKARPS6KB1AURKBPARP1PARP2
SCHEMBL7251899 0.83 AURKA (0.48) AURKARPS6KB1AURKBPARP1PARP2
SCHEMBL484230 0.83 AURKA (0.48) AURKARPS6KB1AURKBPARP1PARP2
Urea SCHEMBL2359624 0.77 HTT (0.42) TAS1R3TAS1R1TAS1R2HAO1ALDH1A1
SCHEMBL11696770 0.75 IDO1 (0.51) HAO1ALDH1A1MAPK1MAPK14GID4
SCHEMBL5349047 0.75 HTR1A (0.44) AURKARPS6KB1AURKBPARP1
SCHEMBL3460627 0.74 PIN1 (0.49) AURKARPS6KB1AURKBPARP1PARP2
SCHEMBL3462221 0.74 PIN1 (0.49) AURKARPS6KB1AURKBPARP1PARP2
SCHEMBL2798590 0.74 PIN1 (0.49) AURKARPS6KB1AURKBPARP1PARP2
SCHEMBL15518445 0.73 HAO1 (0.51) TAS1R3TAS1R1TAS1R2HAO1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999052857-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 1999-10-21 WO disclosed