SCHEMBL7252122

SCHEMBL7252122

O=C(c1cccc(O)c1)N1CCNCC1

nearest known ligand 0.74

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.67
MGLL Q99685 8/20 0.58
GABRD O14764 1/20 0.52
GABRA1 P14867 1/20 0.52
GABRB1 P18505 1/20 0.52
GABRA5 P31644 1/20 0.52
GABRA3 P34903 1/20 0.52
GABRA2 P47869 1/20 0.52
GABRB2 P47870 1/20 0.52
GABRA4 P48169 1/20 0.52
PARP1 P09874 1/20 0.52
ALDH1A1 P00352 1/20 0.51
TP53 P04637 1/20 0.51
HRH4 Q9H3N8 1/20 0.50
HRH3 Q9Y5N1 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8358286 0.90 SIGMAR1 (0.76) SIGMAR1GABRDGABRA1GABRB1GABRA5
SCHEMBL3584183 0.85 SIGMAR1 (0.69) SIGMAR1GABRDGABRA1GABRB1GABRA5
SCHEMBL2644377 0.84 HPGD (0.67) MGLLALDH1A1TP53
SCHEMBL15605882 0.84 SMN1; SMN2 (0.65) MGLLALDH1A1TP53
SCHEMBL20267190 0.83 SIGMAR1 (0.72) SIGMAR1GABRDGABRA1GABRB1GABRA5
SCHEMBL4053730 0.83 HPGD (0.68) MGLLALDH1A1
SCHEMBL4053727 0.83 HPGD (0.68) MGLLALDH1A1
SCHEMBL30957287 0.83 HPGD (0.68) MGLLALDH1A1
SCHEMBL2336862 0.82 SMN1; SMN2 (0.71) SIGMAR1ALDH1A1
SCHEMBL14107680 0.82 SIGMAR1 (0.65) SIGMAR1MGLLGABRDGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102898377-A Novel phthalazinone derivatives and uses thereof NANJING SANHOME PHARMACEUTICAL CO LTD 2013-01-30 CN disclosed
US-6512000-B1 Aminocarbonyl- substituted benzimidazole derivatives for the treatment of diseases in which inhibition of tryptase is of therapeutic such as for treating an inflammatory or allergic disease BOEHRINGER INGELHEIM PHARMA KG (DE) 2003-01-28 US disclosed