SCHEMBL7253276

SCHEMBL7253276

CN(C)CCn1ccc2ccc(N3CCOCC3)cc21

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 9/20 0.61
HTR2A P28223 3/20 0.53
HTR2C P28335 3/20 0.53
PIK3CA P42336 3/20 0.46
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
MAPK1 P28482 1/20 0.45
HTR6 P50406 1/20 0.42
GRM2 Q14416 1/20 0.41
NOS3 P29474 2/20 0.41
NOS1 P29475 2/20 0.41
MTOR P42345 1/20 0.41
NOS2 P35228 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7253044 0.85 HTR1D (0.61) HTR1DHTR2AHTR2CHTR6NOS3
SCHEMBL7988144 0.79 MAPT (0.42) HTR1DUSP2ALDH1A1LMNAPOLB
SCHEMBL7253617 0.78 HTR1D (0.51) HTR1DHTR2AHTR2CHTR6NOS3
SCHEMBL7527390 0.78 MAPT (0.48) PIK3CAUSP2ALDH1A1LMNAPOLB
SCHEMBL7253095 0.78 CDK8 (0.41) HTR1DPIK3CAALDH1A1LMNAMAPT
SCHEMBL7253663 0.76 HTR1D (1.00) HTR1DHTR2AHTR2CHTR6NOS3
SCHEMBL7804940 0.75 HTR2C (0.57) HTR1DHTR2AHTR2CHTR6NOS3
SCHEMBL7253250 0.74 HTR1D (1.00) HTR1DHTR2AHTR2CHTR6NOS3
Hydrochloric Acid SCHEMBL8035287 0.74 HTR2C (0.56) HTR1DHTR2AHTR2CHTR6NOS3
SCHEMBL7994198 0.73 RAB9A (0.52) ALDH1A1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020169322-A1 Use of N-alkylamino-heterocylic compounds for the treatment of migraine NPS ALLEXLIX CORP. 2002-11-14 US claimed
US-6635639-B2 Treatment or diagnosis of central nervous system conditions NPS ALLELIX CORP. (CA) 2003-10-21 US disclosed
US-20020169322-A1 Use of N-alkylamino-heterocylic compounds for the treatment of migraine NPS ALLEXLIX CORP. 2002-11-14 US disclosed
US-6380242-B1 FOR DIAGNOSIS AND THERAPY OF CENTRAL NERVOUS SYSTEM CONDITIONS NPS ALLELIX CORP. (CA) 2002-04-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020169322-A1 Use of N-alkylamino-heterocylic compounds for the treatment of migraine CNR1, CNR2, KCNH1 HTR1D 128/4885HTR2A 425/4885HTR2C 127/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.